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| 产品编号 | 包装单位 | 单价(元) | 国内现货 | 国外库存 | 询价单 |
| 3088218 | 10 MG | 2310 | |||
| 3088218 | 50 MG | 6710 |
产品别名
1841-19-6
Fluspirilene
8-[4,4-bis(p-Fluorophenyl)butyl]-1-phenyl-1,3,8-triazino[4.5]decan-4-one
R 6218
结构式
基本信息
| Empirical Formula【经验(实验)分子式】 | C29H31F2N3O |
| Molecular weight | 475.57 |
| EC number【EC 号】 | 217-418-6 |
| MDL number | MFCD00055137 |
| PubChem Substance ID【PubChem化学物质编号】 | 24277915 |
| NACRES | NA.77 |
| Application【应用】 | Fluspirilene has been used as a neuroleptic drug to study its effects on human ether-a-go-go related gene (HERG). Fluspirilene has been used to study its cytotoxicity effect on malignant glioma. |
| Biochem/physiol Actions【生化/生理作用】 | Fluspirilene has a potential to inhibit the activity of cyclin-dependent kinase 2 (CDK2). It is an effective anti-cancer agent used for treating human hepatocellular carcinoma. Fluspirilene is a dopamine receptor antagonist. It also acts as a calcium channel blocker. Fluspirilene is an antipsychotic agent and exhibits neuoleptic properties. It exhibits therapeutic effects against glioblastoma and Schizophrenia. |
| Features and Benefits【特点和优势】 | This compound was developed by Johnson & Johnson. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here. |
产品性质
| Assay【测定】 | ≥98% (HPLC) |
| form【形式】 | solid |
| color【颜色】 | white |
| solubility【溶解性】 | DMSO: ≥20 mg/mL H2O: insoluble ethanol: soluble |
| originator【创始人】 | Johnson & Johnson |
| storage temp.【储存温度】 | room temp |
| SMILES string | Fc1ccc(cc1)C(CCCN2CCC3(CC2)N(CNC3=O)c4ccccc4)c5ccc(F)cc5 |
| InChI | 1S/C29H31F2N3O/c30-24-12-8-22(9-13-24)27(23-10-14-25(31)15-11-23)7-4-18-33-19-16-29(17-20-33)28(35)32-21-34(29)26-5-2-1-3-6-26/h1-3,5-6,8-15,27H,4,7,16-21H2,(H,32,35) |
| InChI key | QOYHHIBFXOOADH-UHFFFAOYSA-N |
| Gene Information | human ... DRD1(1812), DRD2(1813), DRD3(1814), DRD4(1815), DRD5(1816) |
| packaging【包装】 | 10, 50 mg in glass bottle |
安全信息
| Storage Class Code【储存分类代码】 | 13 - Non Combustible Solids |
| WGK | WGK 3 |
| Personal Protective Equipment【个人防护装备】 | Eyeshields, Gloves, type N95 (US) |
