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Tegaserod maleate
产品价格查看更多规格...
产品编号 | 包装单位 | 单价(元) | 国内现货 | 国外库存 | 询价单 |
3248980 | 10 MG | 1380 | |||
3248980 | 50 MG | 5070 |
产品别名
189188-57-6
Tegaserod maleate
2-[(5-Methoxy-1H-indol-3-yl)methylene]-N-pentyl-hydrazinecarboximidamide maleate
结构式
基本信息
Empirical Formula【经验(实验)分子式】 | C16H23N5O · C4H4O4 |
Molecular weight | 417.46 |
MDL number | MFCD09028009 |
PubChem Substance ID【PubChem化学物质编号】 | 329825925 |
NACRES | NA.77 |
Application【应用】 | Tegaserod maleate has been used to study its cytotoxic effects on human astrocytes and to study its effects as an anti-glioblastoma agent. |
Biochem/physiol Actions【生化/生理作用】 | It stimulates neurotransmitter release from enteric nerves and regularizes gastrointestinal function. Tegaserod has been used to treat irritable bowel syndrome associated with constipation and chronic constipation. Tegaserod is a potent full agonist at serotonin 5-HT4 receptors with an EC50 of 7 nM. |
产品性质
Quality Level【质量水平】 | 100 |
Assay【测定】 | ≥98% (HPLC) |
form【形式】 | powder |
color【颜色】 | white to beige |
solubility【溶解性】 | DMSO: 20 mg/mL, clear |
storage temp.【储存温度】 | 2-8℃ |
SMILES string | N=C(NCCCCC)N/N=C/C1=CNC2=C1C=C(OC)C=C2.OC(/C=C\C(O)=O)=O |
InChI | 1S/C16H23N5O.C4H4O4/c1-3-4-5-8-18-16(17)21-20-11-12-10-19-15-7-6-13(22-2)9-14(12)15;5-3(6)1-2-4(7)8/h6-7,9-11,19H,3-5,8H2,1-2H3,(H3,17,18,21);1-2H,(H,5,6)(H,7,8)/b20-11+;2-1- |
InChI key | CPDDZSSEAVLMRY-FEQFWAPWSA-N |
Gene Information | human ... HTR4(3360) |
packaging【包装】 | 10, 50 mg in glass bottle |
安全信息
Storage Class Code【储存分类代码】 | 13 - Non Combustible Solids |
WGK | WGK 3 |