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CGS-9343B
产品编号: | 3424631 |
规格: | ≥98% (HPLC), powder |
CAS NO: | 109826-27-9 |
包装规格: | 5 MG,25 MG |
产品类别: | 进口试剂 |
品牌: | Sigma-Aldrich |
优惠价: | 立即咨询 |
产品别名
109826-27-9
CGS-9343B
Zaldaride maleate
CGS9343B
1,3-Dihydro-1-[1-[(4-methyl-4H,6H-pyrrolo[1,2-a][4,1]- benzoxazepin-4-yl)methyl]-4-piperidinyl]-2H-benzimidazol-2-one maleate
KW-5617
结构式
基本信息
Empirical Formula【经验(实验)分子式】 | C26H28N4O2 · C4H4O4 |
Molecular weight | 544.60 |
MDL number | MFCD04113002 |
PubChem Substance ID【PubChem化学物质编号】 | 329774899 |
NACRES | NA.77 |
Biochem/physiol Actions【生化/生理作用】 | CGS-9343B is a selective calmodulin antagonist with minimal protein kinase C or antidopaminergic activity. CGS-9343B is a potent inhibitor of calmodulin-activated (Type I) phosphodiesterase activity with IC50 in the nanomolar range. |
Features and Benefits【特点和优势】 | This compound was developed by Novartis. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here. |
产品性质
Quality Level【质量水平】 | 100 |
Assay【测定】 | ≥98% (HPLC) |
form【形式】 | powder |
color【颜色】 | white to off-white |
solubility【溶解性】 | DMSO: >10 mg/mL |
originator【创始人】 | Novartis |
storage temp.【储存温度】 | 2-8℃ |
SMILES string | OC(=O)\C=C/C(O)=O.CC4(CN1CCC(CC1)N2C(=O)Nc3ccccc23)OCc5ccccc5-n6cccc46 |
InChI | 1S/C26H28N4O2.C4H4O4/c1-26(24-11-6-14-29(24)22-9-4-2-7-19(22)17-32-26)18-28-15-12-20(13-16-28)30-23-10-5-3-8-21(23)27-25(30)31;5-3(6)1-2-4(7)8/h2-11,14,20H,12-13,15-18H2,1H3,(H,27,31);1-2H,(H,5,6)(H,7,8)/b;2-1- |
InChI key | NGODOSILXOFQPH-BTJKTKAUSA-N |
packaging【包装】 | 5, 25 mg in glass bottle |
安全信息
Storage Class Code【储存分类代码】 | 11 - Combustible Solids |
WGK | WGK 3 |